Enzyme inhibitors are often designed to mimic the transition state or intermediate of an enzyme-catalyzed reaction.
Bewertung:The mechanism of orthosteric inhibition is simply to prevent substrate binding to the enzyme through direct competition which in turn prevents the enzyme from catalysing the conversion of substrates into products.
Bewertung:H-89 is a protein kinase inhibitor with greatest effect on protein kinase A.
Bewertung:Qnz inhibitor is a common feature of metabolic pathway control in cells.
Bewertung:Liproxstatin-1 is an effective inhibitor of oligodendrocyte ferroptosis
Bewertung:pf-00299804 inhibitor is a medication for the treatment of non-small-cell lung carcinoma.
Bewertung:This gene belongs to the protein kinase superfamily.
Bewertung:A high specificity and potency ensure that a drug will have few side effects and thus low toxicity.
Bewertung:mTOR inhibitors are a class of drugs that inhibit the mechanistic target of rapamycin.
Bewertung:Other artificial enzyme inhibitors block acetylcholinesterase, an enzyme which breaks down acetylcholine, and are used as nerve agents in chemical warfare.
Bewertung:Epirubicin inhibitor generates free radicals that cause cell and DNA damage.
Bewertung:The transmembrane transporters inhibitors are a transport system superfamily that is one of the largest and possibly one of the oldest gene families.
Bewertung:Sc75741 inhibitor form a chemical bond with the enzyme such that the enzyme is inhibited until the chemical bond is broken.
Bewertung:BV6 inhibits the cell viability of HCC193 NSCLC cells with IC50 of 7.2 μM
Bewertung:Although the trypsin inhibitor is a protein, it avoids being hydrolysed as a substrate by the protease by excluding water from trypsin's active site and destabilising the transition state.
Bewertung:GW-572016 inhibitor is an orally active drug for breast cancer and other solid tumours.
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Bewertung:Viagra is classified as a phosphodiesterase type 5 (PDE5) inhibitor. Viagra (sildenafil) is a brand-name oral tablet prescribed for erectile dysfunction. The main differences are cost and timing. For occasional use, most people start with Viagra which ..
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